This is a list of opioids, opioid antagonists and inverse agonists.
Polish heroin (Compote, Kompot) • Diascordium • B & O Supprettes • Dover's powder • Kendal Black Drop • Laudanum • Mithridate • Opium • Paregoric • Poppy straw concentrate • Poppy tea • Smoking opium • Theriac
Codeine • Morphine • Oripavine • Pseudomorphine • Thebaine
Pantopon • Papaveretum (Omnopon) • Tetrapon
14-Hydroxymorphine • 2,4-Dinitrophenylmorphine • 6-Methyldihydromorphine • 6-Methylenedihydrodesoxymorphine • 6-Acetyldihydromorphine • Azidomorphine • Chlornaltrexamine • Chloroxymorphamine • Desomorphine (dihydrodesoxymorphine) • Dihydromorphine • Ethyldihydromorphine • Hydromorphinol • Methyldesorphine • N-Phenethylnormorphine • RAM-378
6-nicotinoyldihydromorphine (Metabolite of Nicomorphine)• Acetylpropionylmorphine • Diacetyldihydromorphine (dihydroheroin, acetylmorphinol) • Dibutyrylmorphine • Dibenzoylmorphine • Diformylmorphine • Dipropanoylmorphine • Heroin (diacetylmorphine) • Nicomorphine •
6-Monoacetylcodeine • Benzylmorphine • Codeine methylbromide • Desocodeine • Dimethylmorphine (methocodeine) • Ethyldihydromorphine • Methyldihydromorphine (dihydroheterocodeine) • Ethylmorphine (dionine) • Heterocodeine • Isocodeine • Pholcodine (morpholinylethylmorphine) • Myrophine • Nalodeine (N-allyl-norcodeine) • Transisocodeine
14-Cinnamoyloxycodeinone • 14-Ethoxymetopon • 14-Methoxymetopon • 14-Phenylpropoxymetopon • 7-Spiroindanyloxymorphone • 8,14-Dihydroxydihydromorphinone • Acetylcodone • Acetylmorphone • α-hydrocodol (=Dihydrocodein, )• Bromoisopropropyldihydromorphinone • Codeinone • Codorphone • Codol (= Codeine Phosphate[1], )• Codoxime • IBNtxA • Thebacon (acetyldihydrocodeinone, dihydrocodeinone enol acetate) • Hydrocodone • Hydromorphone • Hydroxycodeine • Metopon (=Methyldihydromorphinone)• Morphenol • Morphinone • Morphol • N-Phenethyl-14-ethoxymetopon • Oxycodone • Oxymorphol • Oxymorphone • Pentamorphone • Semorphone
α-chlorocodide (= Chlorocodide) • β-chlorocodide • α-chloromorphide (= Chloromorphide)• Bromocodide • Bromomorphide • Chlorodihydrocodide • Chloromorphide • Codide
14-Hydroxydihydrocodeine • Acetyldihydrocodeine • Dihydrocodeine • Dihydrodesoxycodeine (desocodeine) • Dihydroisocodeine • Nicocodeine • Nicodicodeine
1-Nitrocodeine cas? [2]• Codeine-N-oxide • Morphine-N-oxide
1-Bromocodeine • 1-Chlorocodeine • 1-Iodomorphine •
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Codeine-N-oxide (genocodeine) • Heroin-7,8-oxide • Morphine-6-glucuronide • 6-Monoacetylmorphine • Morphine-N-oxide (genomorphine) • Naltrexol • Norcodeine • Normorphine
Cyclorphan • Dextrallorphan • Levorphanol • Levophenacylmorphan • Levomethorphan • Norlevorphanol • Oxilorphan • Phenomorphan • Methorphan (racemethorphan) • Morphanol (racemorphanol) • Ro4-1539 • Xorphanol
Butorphanol • Cyprodime • Drotebanol • Fenfangjine G • Nalbuphine • Sinomenine (cocculine) •
5,9 alpha-diethyl-2-hydroxybenzomorphan (5,9-DEHB) • 8-Carboxamidocyclazocine (8-CAC) • Alazocine • Anazocine • Bremazocine • Butinazocine • Carbazocine • Cogazocine • Cyclazocine • Dezocine • Eptazocine • Etazocine • Ethylketocyclazocine • Fedotozine Fluorophen • Gemazocine • Ibazocine • Ketazocine • Metazocine • Moxazocine • Pentazocine • Phenazocine • Quadazocine • Streptozocine • Thiazocine • Tonazocine • Volazocine • Zenazocine
4-Fluoromeperidine • Allylnorpethidine • Anileridine • Benzethidine • Carperidine • Difenoxin • Diphenoxylate • Etoxeridine (carbetidine) • Furethidine • Hydroxypethidine (bemidone) • Morpheridine • Oxpheneridine (carbamethidine) • Meperidine-N-oxide • Pethidine (meperidine) • Pethidine intermediate A • Pethidine intermediate B (norpethidine) • Pethidine intermediate C (pethidinic acid) • Pheneridine • Phenoperidine • Piminodine • Properidine (ipropethidine) • Sameridine
Allylprodine • (α/β)-Meprodine • Desmethylprodine (MPPP) • PEPAP • (α/β)-Prodine • Prosidol • Trimeperidine (promedol)
Acetoxyketobemidone • Droxypropine • Ketobemidone • Methylketobemidone • Propylketobemidone
Alvimopan • Loperamide • Picenadol
Dextromethadone • Dipipanone • Isomethadone • Levoisomethadone • Levomethadone • Methadone • Methadone intermediate [3]• Normethadone • Norpipanone • Phenadoxone (heptazone) • Pipidone (3-hexanone,6-piperidino-4,4-diphenyl-5-methyl) [4]
Alphaacetylmethadol • Dimepheptanol (racemethadol) • Levacetylmethadol • Noracetylmethadol
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Desmethylmoramide • Dextromoramide • Levomoramide • Moramide intermediate [5]• Racemoramide
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Diethylthiambutene • Dimethylthiambutene • Ethylmethylthiambutene • Piperidylthiambutene • Pyrrolidinylthiambutene • Thiambutene • Tipepidine
Dextropropoxyphene (propoxyphene) • Dimenoxadol • Dioxaphetyl butyrate • Levopropoxyphene • Norpropoxyphene
Diampromide • Phenampromide • Propiram
IC-26 • Isoaminile • Lefetamine • R-4066
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3-Allylfentanyl • 3-Methylfentanyl • 3-Methylthiofentanyl • 4-Phenylfentanyl • Alfentanil • Alphamethylacetylfentanyl • Alphamethylfentanyl • Alphamethylthiofentanyl • Benzylfentanyl [6] • Betahydroxyfentanyl • Betahydroxythiofentanyl • Betamethylfentanyl • Brifentanil • Carfentanil • Fentanyl • Lofentanil • Mirfentanil • Ocfentanil • Ohmefentanyl • Parafluorofentanyl • Phenaridine • Remifentanil • Sufentanil • Thenylfentanyl [7]• Thiofentanyl • Trefentanil
7-PET • Acetorphine • Alletorphine (N-allyl-noretorphine) • BU-48 • Buprenorphine • Cyprenorphine • Dihydroetorphine • Etorphine • Homprenorphine • 18,19-Dehydrobuprenorphine (HS-599) [8] [9]• N-cyclopropylmethylnoretorphine [10]• Nepenthone • Norbuprenorphine • Thevinone [11] • Thienorphine [12]
Ethoheptazine • Meptazinol • Metheptazine • Metethoheptazine • Proheptazine
Clonitazene • Etonitazene • Nitazene
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18-Methoxycoronaridine • 7-Acetoxymitragynine • 7-Hydroxymitragynine • Akuammidine • Akuammine • Eseroline • Hodgkinsine • Mitragynine • Pericine • Pseudoakuammigine
BW373U86 • DPI-221 • DPI-287 • DPI-3290 • SNC-80
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Big dynorphin • Dynorphin A • Dynorphin B
Beta-endorphin • Alpha-endorphin • Gamma-endorphin • α-neo-endorphin • β-neo-endorphin
DADLE • DAMGO • Dermenkephalin • Met-enkephalin • Leu-enkephalin
Adrenorphin • Amidorphin • Casomorphin • DALDA • Deltorphin • Dermorphin • DPDPE • Endomorphin • Gliadorphin • Morphiceptin • Nociceptin • Octreotide • Opiorphin • Rubiscolin • TRIMU 5
3-(3-Methoxyphenyl)-3-ethoxycarbonyltropane • AD-1211 • AH-7921 • Azaprocin • BDPC • Bisnortilidine [13] [14] • BRL-52537 • Bromadoline • C-8813 • Ciramadol • Doxpicomine • Enadoline • Faxeladol • GR-89696 • Herkinorin • ICI-199,441 • ICI-204,448 • J-113,397 • JTC-801 • Ketamine • KNT-42 • LPK-26 • Methopholine • MT-45 • Desmethylclozapine • NNC 63-0532 • Nortilidine • O-Desmethyltramadol • Phenadone • Phencyclidine • Prodilidine • Profadol • Ro64-6198 • Salvinorin A • SB-612,111 • SC-17599 • RWJ-394,674 • TAN-67 • Tapentadol • Tecodine=Oxycodone [15] • Tifluadom • Tilidine • Tramadol • Trimebutine • U-50,488 • U-69,593 • Viminol • 1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide (W-18)
5'-Guanidinonaltrindole • β-Funaltrexamine • 6β-Naltrexol • Alvimopan • Binaltorphimine • Chlornaltrexamine • Clocinnamox • Cyclazocine • Cyprodime • Diacetylnalorphine [16] • Difenamizole [17]• Diprenorphine (M5050) • Fedotozine • JDTic • Levallorphan • Methocinnamox • Methylnaltrexone • Nalfurafine • Nalmefene • Nalmexone [18] • Naloxazone • Naloxonazine • Naloxone • Naloxone benzoylhydrazone • Nalorphine • Naltrexone • Naltriben • Naltrindole • Norbinaltorphimine • Oxilorphan • S-allyl-3-hydroxy-17-thioniamorphinan (SAHTM)[19]